From: Branched-chain amino acid aminotransferase and methionine formation in Mycobacterium tuberculosis
Inhibitor | Kic(μM) | Kiu(μM) |
---|---|---|
O-(t-butyl)hydroxylamine | 11.02 ± 2.76 | 85.60 ± 44.79 |
carboxymethoxylamine | 20.97 ± 7.27 | 142.42 ± 69.76 |
O-allylhydroxylamine | 21.61 ± 11.08 | >200 (386)* |
O-benzylhydroxylamine | 8.20 ± 2.56 | 84.08 ± 31.91 |